Tolifast SR 450mg Tablets 6′

Description

Tolifast SR 450mg is a medication that contains Tolperisone Hydrochloride as its active ingredient. It is typically used as a muscle relaxant to treat conditions involving muscle spasm or stiffness. The SR in the name stands for Sustained Release, meaning the medication is released slowly into the bloodstream to provide prolonged effects.

Active Ingredient:

• Tolperisone Hydrochloride 450 mg (Sustained Release)

Uses of Tolifast SR 450mg:

Tolperisone is primarily used to relieve muscle spasms and to treat certain neurological disorders that cause muscle stiffness and discomfort. Its uses include:

1. Muscle Spasms:
   • Tolperisone is commonly used to treat acute muscle spasms associated with conditions like musculoskeletal pain, back pain, or neck pain.
2. Neurological Disorders:
   • It is also used for conditions that involve muscle spasticity due to neurological disorders like multiple sclerosis (MS), cerebral palsy, stroke, or spinal cord injuries. These conditions often cause stiff or rigid muscles, which Tolperisone helps to relieve.
3. Post-Surgical Muscle Spasms:
   • After surgery, especially orthopedic or spinal surgeries, patients may experience muscle spasms. Tolperisone can be prescribed to reduce this discomfort.
4. Fibromyalgia:
   • Some people with fibromyalgia, a chronic condition that causes widespread muscle pain, may benefit from Tolperisone’s muscle-relaxing effects.

How Tolifast SR 450mg Works:

Tolperisone is a central muscle relaxant. It works by inhibiting the signals that cause muscles to contract, helping to reduce muscle tension and muscle stiffness.

• Central action: Tolperisone works on the central nervous system (CNS) to block the transmission of nerve signals that lead to muscle contraction. By doing so, it reduces the intensity and frequency of muscle spasms.
• Sustained release formulation (SR): The sustained release formulation allows Tolperisone to be released gradually into the body over an extended period. This provides more consistent relief and can help minimize the need for frequent doses.

Dosage and Administration:

The dosage of Tolifast SR 450mg will depend on the condition being treated and the patient’s response to the medication. The sustained-release formulation typically means the medication is taken once a day, but you should always follow your doctor’s instructions.

• Usual Dose:
  • For adults: The typical starting dose is 450 mg once daily, usually taken with a glass of water. The dose may be adjusted by your healthcare provider based on your individual response and the severity of your condition.
  • For elderly patients: A lower dose may be recommended for elderly individuals or those with impaired liver or kidney function.
  • Missed dose: If you miss a dose, take it as soon as you remember, unless it’s almost time for the next dose. Do not take two doses to make up for a missed dose.
• Administration:
  • Take with water: Swallow the tablet whole with a glass of water. Do not crush, chew, or break the tablet, as this could affect how the medication is absorbed.
  • Food: Tolifast can typically be taken with or without food, but it’s always best to follow your doctor’s specific instructions.

Side Effects of Tolifast SR 450mg:

Tolperisone is generally well tolerated, but like all medications, it may cause some side effects. Some common and serious side effects include:

1. Common Side Effects:
   • Drowsiness or sedation
   • Dizziness or lightheadedness
   • Headache
   • Nausea or stomach discomfort
   • Fatigue
   • Gastrointestinal issues (e.g., diarrhea, constipation)
   • Dry mouth
   • Muscle weakness
2. Serious Side Effects (Rare):
   • Severe allergic reactions: Symptoms such as swelling of the face, lips, or tongue, difficulty breathing, or hives (urticaria) should be treated as a medical emergency.
   • Liver or kidney problems: Symptoms may include yellowing of the skin or eyes (jaundice), dark urine, or abdominal pain.
   • Severe dizziness or fainting: Especially if standing up suddenly, as Tolperisone may cause a drop in blood pressure.
   • Severe muscle weakness: In some cases, the medication can exacerbate muscle weakness, especially in people with certain underlying conditions.
3. Overdose:
   • An overdose of Tolperisone can cause extreme drowsiness, nausea, vomiting, and respiratory depression. Seek immediate medical attention if an overdose is suspected.

Precautions and Warnings:

• Drowsiness: Tolperisone can cause drowsiness or dizziness, so be cautious when driving, operating machinery, or performing tasks that require full concentration.
• Kidney or Liver Disease: If you have a history of liver or kidney disease, your doctor may adjust the dose of Tolperisone or monitor your liver and kidney function closely during treatment.
• Alcohol: Alcohol can increase the sedative effects of Tolperisone, leading to increased drowsiness or dizziness. It’s advisable to limit alcohol consumption while taking this medication.
• Pregnancy and Breastfeeding: The safety of Tolperisone during pregnancy and breastfeeding has not been fully established, so it should be used only if the potential benefits outweigh the risks. Consult your doctor if you are pregnant or breastfeeding.
• Elderly: Older adults may be more sensitive to the side effects of Tolperisone, particularly dizziness and drowsiness. Lower doses may be recommended.

Drug Interactions:

Tolperisone may interact with other medications, so it’s important to inform your healthcare provider about all other medications you are currently taking, including over-the-counter drugs and herbal supplements.

1. CNS Depressants: Combining Tolperisone with other CNS depressants (e.g., sedatives, antihistamines, alcohol) may increase the risk of excessive drowsiness or sedation.
2. Antihypertensive Medications: If you are on blood pressure-lowering medications, Tolperisone may enhance the blood pressure-lowering effects, potentially leading to dizziness or fainting.
3. Other Muscle Relaxants: Caution should be exercised when combining Tolperisone with other muscle relaxants, as the sedative effects may be amplified.

Storage:

• Tolifast SR 450mg should be stored at room temperature (between 15°C and 30°C), away from moisture, heat, and direct sunlight.
• Keep the medication in its original packaging and out of reach of children.
• Do not use the medication past its expiration date.